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Panduan penyiapan dan pemberian terapi medikasi
Ceftriaxone

Penyiapan

Sediaan

  • 250mg
  • 500mg
  • 1gr
  • 2gr

Rekomendasi Pengenceran (Konsentrasi)

  • injeksi IV: 10-40mg/ml (250mg dalam 6,25cc, 500mg dalam 12,5cc, 1gr dalam 25cc, 2gr dalam 50cc)
  • injeksi IM: 250 dalam 1ml, 500mg dalam 2cc, 1gr dalam 4cc, 2gr dalam 7,5cc

Pelarut

  • D5%
  • NaCl 0.9%
  • RL
  • WI

Pemberian

Rekomendasi Akses

IV
IM

Rekomendasi Durasi Pemberian

intermiten dalam 15-30menit

Stabilitas Obat Setelah Rekonstruksi

24 jam dalam suhu 25C

Keamanan

pH

6,7
pH risiko rendah (5,0-7,5)

Osmolaritas Sesudah Pengenceran

konsentrasi 50mg/ml dalam NS 0,9% = 364mOsm/kg
Osmolaritas rendah (<600)

Phlebitis

Tidak

Inkompatibilitas

  • Aminophylline
  • Calcium chloride
  • Calcium gluconate
  • Clindamycin phosphate
  • Gentamicin sulfate
  • Linezolid
  • Theophylline,
  • Lidocaine HCl
  • Amsacrine
  • Anakinra
  • Azithromycin
  • Caspofungin acetate
  • Filgrastim
  • Fluconazole
  • Isavuconazium sulfate
  • Lebetalol HCl
  • Pentamidine isethionate
  • Vancomycin HCl
  • Vinorelbine tartate

Klasifikasi GHS

Irritant
Health Hazard

Manifestasi GHS

315 (100%): Causes skin irritation [Warning Skin corrosion/irritation]
H317 (100%): May cause an allergic skin reaction [Warning Sensitization, Skin]
H319 (100%): Causes serious eye irritation [Warning Serious eye damage/eye irritation]
H334 (100%): May cause allergy or asthma symptoms or breathing difficulties if inhaled [Danger Sensitization, respiratory]
H335 (100%): May cause respiratory irritation [Warning Specific target organ toxicity, single exposure; Respiratory tract irritation]

Sumber

  • American Society of Health-System Pharmacists. 2021. ASHP® Injectable Drug Information: A Comprehensive Guide to Compatibility and Stability. 2021 Edition. eBook. American Society of Health-System Pharmacists. ISBN: 978-1-58528-690-4. doi.org/10.37573/9781585286850
  • https://pubchem.ncbi.nlm.nih.gov/compound/5479530