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Panduan penyiapan dan pemberian terapi medikasi
Fluconazole

Penyiapan

Sediaan

  • 200 mg/100 mL

Rekomendasi Pengenceran (Konsentrasi)

tidak diencerkan

Pelarut

Pemberian

Rekomendasi Akses

IV

Rekomendasi Durasi Pemberian

200 mg/jam

Stabilitas Obat Setelah Rekonstruksi

Keamanan

pH

4,0-6,5
pH risiko sedang (4,0-5,0 / 7,5-9,0)

Osmolaritas Sebelum Pengenceran

300-315
Osmolaritas rendah (<600)

Phlebitis

Tidak

Inkompatibilitas

  • Trimethoprim Sulfamethoxazole
  • Pentamidine Isethionate
  • Imipenem Cilastatin Sodium
  • Hydroxyzine HCl
  • Haloperidol Lactate
  • Furosemide
  • Fat Emulsion
  • Digoxin
  • Diazepam
  • Clindamycin Phosphate
  • Chloramphenicol Sodium Succinate
  • Ceftriaxone Sodium
  • Cefuroxime Sodium
  • Ceftazidime
  • Cefotaxime Sodium
  • Ampicillin Sodium

Klasifikasi GHS

Irritant
Health Hazard

Manifestasi GHS

H302 (99.5%): Harmful if swallowed [Warning Acute toxicity, oral]
H315 (68.5%): Causes skin irritation [Warning Skin corrosion/irritation]
H319 (57.4%): Causes serious eye irritation [Warning Serious eye damage/eye irritation]
H335 (29.4%): May cause respiratory irritation [Warning Specific target organ toxicity, single exposure; Respiratory tract irritation]
H360 (54.3%): May damage fertility or the unborn child [Danger Reproductive toxicity]
H362 (47.7%): May cause harm to breast-fed children [Reproductive toxicity, effects on or via lactation]
H371 (31%): May cause damage to organs [Warning Specific target organ toxicity, single exposure]
H412 (46.7%): Harmful to aquatic life with long lasting effects [Hazardous to the aquatic environment, long-term hazard]

Sumber

  • National center for biotechnology information. PubChem Compound Summary for CID 3365, Fluconazole.
  • https://pubchem.ncbi.nlm.gov/compound/Fluconazole.
  • American Society of Health-System Pharmacists. 2021. ASHP® Injectable Drug Information: A Comprehensive Guide to Compatibility and Stability. 2021 Edition. eBook. American Society of Health-System Pharmacists. ISBN: 978-1-58528-690-4. doi.org/10.37573/9781585286850
  • https://pubchem.ncbi.nlm.nih.gov/compound/fluconazole